EPZ-719 is a novel and potent SETD2 inhibitor ( IC50 = 0.005 μM) with a high selectivity over other histone methyltransferases. SET domain-containing protein 2 (SETD2), a histone methyltransferase, has been identified as a target of interest in certain hematological malignancies, including multiple myeloma.

 

Brand: BCM

 

InChi Key: ZLVKIBLQXFILMA-IKGGRYGDSA-N

 

Attribute
[Chem Name]	1H-Indole-2-carboxamide, 4-fluoro-7-methyl-N-[(1R,3S)-3-[(3S)-3-[methyl(methylsulfonyl)amino]-1-pyrrolidinyl]cyclohexyl]-, rel-
[Synonym]	EPZ-719; EPZ 719; EPZ719
[CAS No.]	2411757-44-1
[Formula]	C22H31FN4O3S
[Molecular]	450.57

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