Lidocaine (Alphacaine) is a selective, reverse peripheral histamine H1 receptor agonist with IC50 greater than 32 μM.

Lidocaine is a local anesthetic, also known as Cerocaine, which has replaced procaine in recent years and is widely used in cosmetic plastic surgery for local infiltration anesthesia. It blocks nerve excitation and conduction by inhibiting sodium ion channels in nerve membranes. Its fat solubility, protein binding rate were higher than procaine, strong penetrating ability, quick action, long action time, effect intensity is 4 times of procaine.

 

Brand: BCM

 

Melting Point: 66-69°C

 

Boiling Point: 372.7±52.0 °C at 760 mmHg

 

Flashing Point: 179.2±30.7 °C

 

pKa: 7.88(H2O)(Approximate)

 

Solubility: Soluble in DMSO; soluble in Water; soluble in Ethanol.

 

Attribute
[CAS No.]	137-58-6
[EINECS]	205-302-8
[Formula]	C14H22N2O
[Molecular]	234.34
[Chem Name]	2-(Diethylamino)-N-(2,6-dimethylphenyl)-acetamide
[Synonym]	Lidocaine; Alphacaine
[Form]	White to slightly yellow powder
[Storage]	Sealed in dry. Store at RT
[MDL No.]	MFCD08443609

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