Lintitript is a selective antagonist of CCK1 with EC50s of 6 nM and 200 nM against CCK1 and CCK2. The Ki value for CCK1 is 0.2 nM.

 

Brand: BCM

 

Solubility: Soluble in DMSO.

 

pKa: 4.00±0.10(Predicted)

 

GHS: GHS05, GHS06

 

Isomeric SMILES: C1=CC=C2C(=C1)C=C(N2CC(=O)O)C(=O)NC3=NC(=CS3)C4=CC=CC=C4Cl  

 

InChIKey: ILNRQFBVVQUOLP-UHFFFAOYSA-N  

 

InChI: InChI=1S/C20H14ClN3O3S/c21-14-7-3-2-6-13(14)15-11-28-20(22-15)23-19(27)17-9-12-5-1-4-8-16(12)24(17)10-18(25)26/h1-9,11H,10H2,(H,25,26)(H,22,23,27)

 

Attribute
[Chem Name]	2-[2-[[4-(2-chlorophenyl)-1,3-thiazol-2-yl]carbamoyl]indol-1-yl]acetic acid
[Synonym]	Lintitript; SR 27897; SR27897; SR-27897
[CAS No.]	136381-85-6
[MDL No.]	MFCD21608519
[Formula]	C20H14ClN3O3S
[Molecular]	411.86
[Form]	White to tan powder
[Storage]	Desiccate at +4°C

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