Galunisertib (LY2157299) is an effective TGFβ receptor I (TβRI) inhibitor with IC50 of 56 nM in cell-free tests. Phase 2 over 3.

 

Brand: BCM

 

Melting Point: 241-242°C

 

Flashing Point: 328.162℃ 

 

Solubility: Soluble in DMSO (up to 25 mg/ml)

 

Stability: Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 1 month.

 

Attribute
[Chem Name]	LY2157299
[CAS No.]	700874-72-2
[Formula]	C22H19N5O
[Molecular]	369.42
[Synonym]	4-[5,6-Dihydro-2-(6-methyl-2-pyridinyl)-4H-pyrrolo[1,2-b]pyrazol-3-yl]-6-quinolinecarboxamide
[Form]	White powder
[Storage]	-20°C
[MDL No.]	MFCD12923319

Goods Tag