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R112 is an ATP-competitive Syk kinase inhibitor with a Ki value of 6 nM. R112 inhibits Syk kinase activity with an IC50 value of 226 nM.
Brand: BCM
Solubility: Soluble in DMSO. Insoluble in Water.
InChi Key: TVKGTSHBQZEFEE-UHFFFAOYSA-N
Attribute [Chem Name] R112 [CAS No.] 575474-82-7 [Synonym] R 112 (pharMaceutical)(E)-Elafibranor575474-82-7R112R-112CHEMBL515271 [Formula] C16H13FN4O2 [Molecular] 312.3 [Form] White to off white solid powder
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