KG-501 is a CREB inhibitor that disrupts Creb-dependent transcription (Ki=10 μM) and CREB: CBP interactions (Ki=50 μM). It also disrupts the binding of phosphorylated CREB(Ser-133) to KIX, a Ki of about 90 μM.

 

Solubility: Soluble in DMSO. Insoluble in water.

 

Attribute
[Chem Name]	KG-501 (2-naphthol-AS-E-phosphate)
[CAS No.]	18228-17-6
[Formula]	C17H13ClNO5P
[Molecular]	377.72
[Synonym]	NAPHTHOLAS-EPHOSPHATE;N-(4-chlorophenyl)-3-(phosphonooxy)naphthalene-2-carboxamide;NAPHTHOLAS-E-PHOSPHATE,FORHISTOLOGY;NAPHTHOLAS-EPHOSPHATENAPHTHOLFREE;N-(4-Chlorophenyl)-3-phosphonooxy-2-naphtChemicalbookhalenecarboxamide;[3-[(4-chlorophenyl)carbamoyl]-2-naphthyl]dihydrogenphosphate;kg-501;N-(4-CHLOROPHENYL)-3-(PHOSPHONOOXY)NAPHTHALENE-2-CARBOXAMIDE;KG-501;NASEP;NAPHTHOLAS-EPHOSPHATE;KG501;KG501
[Storage]	Keep in dark place,Inert atmosphere, 2-8°C
[EINECS]	242-106-1
[MDL No.]	MFCD00042718
[Form]	Solid powder

Goods Tag