Name：Picrotoxinin

Catalog No.：
BCM006711

Chem Name：
(1R,3R,5S,8S,9R,12S,13R,14R)-1-hydroxy-13-methyl-14-prop-1-en-2-yl-4,7,10-trioxapentacyclo[6.4.1.19,12.03,5.05,13]tetradecane-6,11-dione

Synonym：
Picrotoxinin; (-)-Picrotoxinin

CAS No.：
17617-45-7

EINECS：
634-009-1

MDL No.：
MFCD00078765

Formula：
C15H16O6

Molecular：
292.28

Form：
Solid

Storage：
Powder: -20°C for 3 years. In solvent: -80°C for 2 years

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SKU	Specification	Brand	Prices	Stock	Cart
BCM006711-25MG	25mg, Purity:98%	BCM	$70	2	Add Cart
BCM006711-50MG	50mg, Purity:98%	BCM	$100	2	Add Cart
BCM006711-100MG	100mg, Purity:98%	BCM	$140	2	Add Cart

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Picrotoxinin is a potent convulsant, a chloride channel blocker. Picrotoxinin is a non-competitive GABAA receptor antagonist that negatively regulates the action of GABA on GABAA receptors. Picrotoxinin inhibits α1β2γ2L GABAA receptors with an IC50 value of 1.15 μM.

Brand: BCM

Target: IC50: 1.15 μM (GABAA receptor)

Melting Point: 203-205°C

pKa: 13.18±0.60(Predicted)

Specific Rotation: D17 +4.4° (c = 4.28 in abs alc), +3.49° (c = 7.57 in acetone)

Solubility: Soluble in DMSO; soluble in Ethanol. Insoluble in Water.

Isomeric SMILES: CC(=C)[C@@H]1[C@@H]2[C@@H]3[C@@]4([C@]([C@H]1C(=O)O2)(C[C@@H]5[C@]4(O5)C(=O)O3)O)C

InChIKey: PIMZUZSSNYHVCU-YKWPQBAZSA-N

InChI: InChI=1S/C15H16O6/c1-5(2)7-8-11(16)19-9(7)10-13(3)14(8,18)4-6-15(13,21-6)12(17)20-10/h6-10,18H,1,4H2,2-3H3/t6-,7+,8-,9-,10-,13-,14-,15+/m1/s1

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[Chem Name] (1R,3R,5S,8S,9R,12S,13R,14R)-1-hydroxy-13-methyl-14-prop-1-en-2-yl-4,7,10-trioxapentacyclo[6.4.1.19,12.03,5.05,13]tetradecane-6,11-dione

[Synonym] Picrotoxinin; (-)-Picrotoxinin

[CAS No.] 17617-45-7

[EINECS] 634-009-1

[MDL No.] MFCD00078765

[Formula] C15H16O6

[Molecular] 292.28

[Form] Solid

[Storage] Powder: -20°C for 3 years. In solvent: -80°C for 2 years

Attribute
[Chem Name]	(1R,3R,5S,8S,9R,12S,13R,14R)-1-hydroxy-13-methyl-14-prop-1-en-2-yl-4,7,10-trioxapentacyclo[6.4.1.19,12.03,5.05,13]tetradecane-6,11-dione
[Synonym]	Picrotoxinin; (-)-Picrotoxinin
[CAS No.]	17617-45-7
[EINECS]	634-009-1
[MDL No.]	MFCD00078765
[Formula]	C15H16O6
[Molecular]	292.28
[Form]	Solid
[Storage]	Powder: -20°C for 3 years. In solvent: -80°C for 2 years